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Drug Agonism

Known as: Agonism, Drug 
Phenomena and pharmaceutics of compounds that selectively bind to a specific receptor and trigger a response. They mimic the action of endogenous… Expand
National Institutes of Health

Papers overview

Semantic Scholar uses AI to extract papers important to this topic.
2015
2015
Type 4 metabotropic glutamate (mGlu4) receptors are emerging targets for the treatment of various disorders. Accordingly… Expand
Highly Cited
2013
Highly Cited
2013
Glucagon, an essential regulator of glucose homeostasis, also modulates lipid metabolism and promotes weight loss, as reflected… Expand
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Highly Cited
2013
Highly Cited
2013
Background—To assess cardiovascular actions of APJ agonism during prolonged (Pyr1)apelin-13 infusion and renin–angiotensin system… Expand
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Review
2012
Review
2012
Abstract  Studies suggest that around 20% of adults in Europe experience chronic pain, which not only has a considerable impact… Expand
Review
2007
Review
2007
  • T. Kenakin
  • Molecular Pharmacology
  • 2007
  • Corpus ID: 5963117
This article describes functional selectivity of agonists and antagonists and distinguishes conventional cell-based functional… Expand
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Highly Cited
2007
Highly Cited
2007
A range of ligands displayed agonism at the long isoform of the human dopamine D2 receptor, whether using receptor-G protein… Expand
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2005
2005
Dexmedetomidine, a highly selective &agr;2-adrenoceptor agonist, is used in combination with local anesthetics for sedation and… Expand
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Highly Cited
2003
Highly Cited
2003
G protein-coupled receptors (GPCRs) are allosteric proteins that adopt inactive (R) and active (R*) conformations in equilibrium… Expand
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2000
2000
Evidence exists for a state of sympathetic hyperactivity in essential hypertension, and moxonidine, a new central sympathetic… Expand
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Review
1996
Review
1996
Sex differences in human responses to nociceptive stimuli and painful pathological conditions have generally indicated that women… Expand