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tropapride

Known as: exo-2,3-dimethoxy-N-(8-(phenylmethyl)-8-azabicyclo(3.2.1)oct-3-yl)benzamide 
National Institutes of Health

Related topics

Related topics

2 relations

Narrower (1)

MD 790501

Broader (1)

Nortropanes

Papers overview

Semantic Scholar uses AI to extract papers important to this topic.
2003
2003
Constitutive Coupling of a Chimeric Dopamine D2/α1 B Receptor to the Phospholipase C Pathway: Inverse Agonism to Silent Antagonism by Neuroleptic Drugs
Neuroleptic drugs have been suggested to act as inverse agonists at the dopamine D2 receptor, but no link between therapeutic… 
2003
2003
Inverse agonism at dopamine D2 receptors: a receptor recalcitrant to high levels of constitutive activation
2001
2001
Dynamic dopamine-antagonist interactions at recombinant human dopamine D(2short) receptor: dopamine-bound versus antagonist-bound receptor states.
Antipsychotic drugs comprise a wide range of structurally diverse compounds and are considered to be antagonists at dopamine D2… 
2001
2001
Atypical kinetics for a series of putative dopamine antagonists to reverse the low-magnitude Ca2+ phase in the dopamine-bound D2short receptor state
Abstract. Real-time analysis of dopamine:antagonist interactions at the recombinant D2short receptor was performed by measuring… 
Highly Cited
1999
Highly Cited
1999
Interactions between neuroleptics and 5-HT1A ligands in preclinical behavioral models for antipsychotic and extrapyramidal effects
Rationale: Combining neuroleptics with 5-HT1A ligands is thought to improve the preclinical profile of neuroleptics and may be of… 
1992
1992
2- and 4-[18F]fluorotropapride, two specific D2 receptor ligands for positron emission tomography: N.C.A. syntheses and animal studies.
1989
1989
Structural requirements of Na+-dependent antidopaminergic agents: Tropapride, Piquindone, Zetidoline, and Metoclopramide Comparison with Na+-independent ligands
SummaryMolecular graphic design coupled with PCILO and crystallographic results have been used to investigate the three… 
1984
1984
Investigation on central dopaminergic receptors (D‐2) using the antagonistic properties of new benzamides
The topography of the central dopaminergic receptor (D−2) has been studied using some analogues of tropapride, a new benzamide… 
1984
1984
Localization of a new benzamide derivative, tropapride and of 1-sulpiride, in the pituitary gland of the rat.
Localization of tropapride and 1-sulpiride in the pituitary gland of the rat has been studied. A comparison of the ratio of total… 
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