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podophyllic acid piperidyl hydrazone nitroxide radical

Known as: PAPHNR 
 
National Institutes of Health

Related topics

Related topics

2 relations
analogs & derivatives

Broader (1)

podofilox

Papers overview

Semantic Scholar uses AI to extract papers important to this topic.
2017
2017
Cholinesterases inhibition and molecular modeling studies of piperidyl-thienyl and 2-pyrazoline derivatives of chalcones.
Super-activation of cholinesterases (acetylcholinesterase and butyrylcholinesterase) are linked to various neurological problems… Expand
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2015
2015
Monoamine Oxidase Inhibition and Molecular Modeling Studies of Piperidyl-thienyl and 2-Pyrazoline Derivatives of Chalcones.
A series of piperidyl-thienyl & 2-pyrazoline derivatives of quinolyl-thienyl chalcones were tested to observe the structural… Expand
2013
2013
Design, synthesis and SAR of piperidyl-oxadiazoles as 11β-hydroxysteroid dehydrogenase 1 inhibitors.
The potential roles of 11β-HSD1 inhibitors in metabolic syndrome, T2D and obesity were well established and currently several… Expand
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2012
2012
Thiorhodamines containing amide and thioamide functionality as inhibitors of the ATP-binding cassette drug transporter P-glycoprotein (ABCB1).
Twelve thiorhodamine derivatives have been examined for their ability to stimulate the ATPase activity of purified human P… Expand
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2011
2011
Anti-HIV-1 and cytotoxicity studies of piperidyl-thienyl chalcones and their 2-pyrazoline derivatives
A series of 12 new pyrazoline derivatives was prepared from piperidyl chalcones, which in turn were synthesized by condensing 4… Expand
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2010
2010
Optimization of piperidyl-ureas as inhibitors of soluble epoxide hydrolase.
Inhibition of sEH is hypothesized to lead to an increase in epoxyeicosatrienoic acids resulting in the potentiation of their anti… Expand
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2002
2002
Antitumor and antioxidant activity of spin labeled derivatives of podophyllotoxin (GP-1) and congeners.
The spin labeled derivative of podophyllotoxin, i.e. podophyllic acid-[4-(2,2,6,6,-tetramethyl-1-piperidyloxy)] hydrazone (GP-1,2… Expand
2002
2002
Exploring the role of bromine at C(10) of (+)-4-[2-[4-(8-chloro-3,10-dibromo- 6,11-dihydro-5H-benzo[5,6]cyclohepta[1,2-b]pyridin-11(R)-yl)-1-piperidinyl]-2- oxoethyl]-1-piperidinecarboxamide (Sch…
The 10-bromobenzocycloheptapyridyl farnesyl transferase inhibitor (FTI) Sch-66336 (1) is currently under clinical evaluation for… Expand
2000
2000
Quantitation of loperamide and N-demethyl-loperamide in human plasma using electrospray ionization with selected reaction ion monitoring liquid chromatography-mass spectrometry.
We report here the development and validation of an LC-MS method for quantitation of loperamide (LOP) and its N-demethyl… Expand
1977
1977
Synthesis and pharmacological properties of a series of antidopaminergic piperidyl benzamides *
The synthesis and pharmacological screening for anti‐apomorphine, stomach emptying and local anaesthetic activities of some new… Expand
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