paullone

 

Topic mentions per year

Topic mentions per year

1999-2017
024619992017

Papers overview

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2010
2010
The reaction of copper(II) chloride or copper(II) acetate with 6-N-(2-N',N'-dimethylaminoethylamino)-7,12-dihydroindolo-[3,2-d][1… (More)
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2006
2006
9-Bromo-7,12-dihydroindolo[3,2-d][1]benzazepin-6(5H)-one, kenpaullone, which displays similarities in the activity profile to… (More)
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2004
2004
With a view to the rational design of selective GSK-3beta inhibitors, 3D-QSAR CoMSIA models were developed for the inhibition of… (More)
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2004
2004
Kenpaullone derivatives with a modified parent ring system were synthesized in order to develop kinase inhibitors with enhanced… (More)
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2003
2003
The majority of human neoplasms have aberrations in the retinoblastoma pathway due to hyperactivation of cyclin-dependent kinases… (More)
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2002
2002
Numerous inhibitors of cyclin-dependent kinases and glycogen synthase kinase-3 (GSK-3) are being developed in view of their… (More)
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2002
2002
Paullones 3 and 4 with aminoalkyl side chains in 2- or 3-position were synthesized as derivatives of kenpaullone 1. Both 3 and 4… (More)
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Highly Cited
2000
Highly Cited
2000
Paullones constitute a new family of benzazepinones with promising antitumoral properties. They were recently described as potent… (More)
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2000
2000
A congeneric series of paullones were characterized using a 3-D QSAR with cyclin-dependent kinase 1 (CDK1) inhibition data. A… (More)
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1999
1999
The paullones represent a novel class of small molecule cyclin-dependent kinase (CDK) inhibitors. To investigate structure… (More)
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