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mesulergine

Known as: N'-(1,6-dimethylergolin-8alpha-yl)-N,N-dimethylsulfamide 
 
National Institutes of Health

Related topics

Related topics

4 relations

Broader (4)

Antiparkinson AgentsDopamine AgonistsErgolinesSerotonin Antagonists

Papers overview

Semantic Scholar uses AI to extract papers important to this topic.
Highly Cited
1995
Highly Cited
1995
(1-(2,5-dimethoxy-4 iodophenyl)-2-aminopropane)-induced head-twitches in the rat are mediated by 5-hydroxytryptamine (5-HT) 2A receptors: modulation by novel 5-HT2A/2C antagonists, D1 antagonists and…
In this study, the involvement of serotonergic and dopaminergic receptors in the modulation of the head-twitch (HTW) response to… Expand
Highly Cited
1993
Highly Cited
1993
Molecular cloning of a mammalian serotonin receptor that activates adenylate cyclase.
Serotonin modulates a wide range of physiological functions by activating multiple receptors, which are coupled to various… Expand
Highly Cited
1993
Highly Cited
1993
A single point mutation (Phe340-->Leu340) of a conserved phenylalanine abolishes 4-[125I]iodo-(2,5-dimethoxy)phenylisopropylamine and [3H]mesulergine but not [3H]ketanserin binding to 5…
The molecular processes by which agonists and antagonists bind to serotonin2 [5-hydroxytryptamine (5-HT2)] receptors are… Expand
Highly Cited
1988
Highly Cited
1988
A nonclassical 5-hydroxytryptamine receptor positively coupled with adenylate cyclase in the central nervous system.
A nonclassical 5-hydroxytryptamine (5-HT) receptor mediates the stimulation of adenylate cyclase activity in mouse embryo… Expand
Highly Cited
1988
Highly Cited
1988
Evidence that mCPP may have behavioural effects mediated by central 5‐HT1C receptors
1 The effects of 1‐(3‐chlorophenyl)piperazine (mCPP) and 1‐[3‐(trifluoromethyl)phenyl] piperazine (TFMPP) on activity of rats in… Expand
Highly Cited
1987
Highly Cited
1987
Characterization of a novel 3H-5-hydroxytryptamine binding site subtype in bovine brain membranes
3H-5-Hydroxytryptamine (5-HT) binding sites were analyzed in bovine brain membranes. The addition of either the 5-HT1A-selective… Expand
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Highly Cited
1986
Highly Cited
1986
Cholinergic terminals in rat hippocampus possess 5-HT1B receptors mediating inhibition of acetylcholine release.
The effects of 5-hydroxytryptamine (5-HT) on the release of [3H]acetylcholine ([3H]ACh) from rat hippocampal nerve endings were… Expand
Highly Cited
1985
Highly Cited
1985
Molecular pharmacology of 5-HT1 and 5-HT2 recognition sites in rat and pig brain membranes: radioligand binding studies with [3H]5-HT, [3H]8-OH-DPAT, (-)[125I]iodocyanopindolol, [3H]mesulergine and…
The pharmacological characteristics of the binding of [3H]8-OH-DPAT ([3H]8-hydroxy-2(di-n-propylamino)tetralin, [125I]CYP… Expand
Highly Cited
1985
Highly Cited
1985
Characterization of the 5-HT1B recognition site in rat brain: binding studies with (-)[125I]iodocyanopindolol.
(-)[125I]Iodocyanopindolol ([125I]CYP) labels rat brain membrane sites which display high affinity for several serotonergic and… Expand
Highly Cited
1984
Highly Cited
1984
Mesulergine, a selective serotonin-2 ligand in the rat cortex, does not label these receptors in porcine and human cortex: evidence for species differences in brain serotonin-2 receptors.
The kinetic and pharmacological characteristics of the binding of [3H]ketanserin and [3H]mesulergine to frontal cortical brain… Expand
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