levocabastine

Known as: Levocabastinum, levocabastine [Chemical/Ingredient], 1-(4-cyano-4-(4-fluorophenyl)cyclohexyl)-3-methyl-4-phenyl-4-piperidinecarboxylic acid 
A synthetic piperidine derivative with antihistamine properties. Levocabastine is a second generation histamine-1 receptor antagonist. When applied… (More)
National Institutes of Health

Papers overview

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2008
2008
Levocabastine is an antiallergic drug acting as a histamine H1-receptor antagonist. In allergic conjunctivitis (AC), it may also… (More)
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1999
1999
The antihistaminic drug levocabastine is a ligand for the low affinity neurotensin receptor (NTS2). Its intracerebroventricular… (More)
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1998
1998
Neurotensin has been shown to produce pharmacological effects both in brain and periphery. Several of these effects are mediated… (More)
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Highly Cited
1996
Highly Cited
1996
This work describes the cloning and expression of the levocabastine-sensitive neurotensin (NT) receptor from mouse brain. The… (More)
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Highly Cited
1996
Highly Cited
1996
A search for sequences homologous to the neurotensin receptor cDNA in a rat hypothalamic library has identified a novel… (More)
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1995
1995
PURPOSE This study was conducted to evaluate the efficacy of 0.05% levocabastine compared with 4% cromolyn for treating allergic… (More)
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Highly Cited
1993
Highly Cited
1993
We describe the characteristics of SR 48692, a selective, nonpeptide antagonist of the neurotensin receptor. In vitro, this… (More)
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1993
1993
Levocabastine is a very potent histamine H1 antagonist, available for ocular use as eye drops containing 0.5 mg/ml of… (More)
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Review
1992
Review
1992
Levocabastine is a new topical histamine H1 antagonist. The antihistaminic and antiallergic effects of levocabastine eye drops… (More)
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1987
1987
Monoiodo-[125I-Tyr3]neurotensin (NT) bound to a high affinity, low capacity binding component and a lower affinity, high capacity… (More)
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