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exaprolol

Known as: 1-isopropylamino-3-(2-cyclohexylphenoxy)-2- propanol 
A lipophilic derivative of the adrenergic blocking agent propranolol with sympatholytic activity. Exaprolol competitively binds to and blocks beta… 
National Institutes of Health

Related topics

Related topics

3 relations

Broader (2)

Adrenergic beta-AntagonistsPropanolamines

Narrower (1)

VULM 456

Papers overview

Semantic Scholar uses AI to extract papers important to this topic.
1991
1991
Effect of chloroquine on isolated mast cells
Chloroquine liberated a relatively low amount of histamine from isolated rat mast cells. In a dose-dependent way, this drug… 
1989
1989
Influence of beta-adrenoceptor blocking drugs on lipid-protein interaction in synaptosomal membranes. An ESR study.
1986
1986
The pharmacokinetics of exaprolol and propranolol in rats with interrupted enterohepatic circulation.
The pharmacokinetics of two beta adrenoceptor blocking drugs, exaprolol and propranolol, in rats with interrupted enterohepatic… 
1985
1985
The interaction of beta-adrenoceptor blocking drugs with platelet aggregation, calcium displacement and fluidization of the membrane.
1985
1985
Exaprolol as a modulator of heart sarcolemmal (Na+ + K+)-ATPase. Evidence for interaction with an essential sulfhydryl group in the catalytic centre of the enzyme.
Beta-adrenoceptor blocking agents may have, in addition to their primary action, also ancillary effects on the cell membrane. In… 
1985
1985
On the interaction of beta-adrenoceptor-blocking drugs with isolated mast cells
The interaction of beta-adrenoceptor blocking drugs (BAB drugs) with isolated mast cells resulted. according to the compound, in… 
1984
1984
Aspects of the cardiovascular pharmacology of exaprolol
This study confirms that exaprolol is a potent β‐adrenoceptor antagonist, having a pA2 value of 9·8 for the inhibition of the… 
1984
1984
Biliary excretion and enterohepatic circulation of two beta-adrenergic blocking drugs, exaprolol and propranolol, in rats.
Plasma levels and excretion of two beta-adrenoceptor blocking drugs 3H-exaprolol and 3H-propranolol were observed up to 96 h… 
1982
1982
Electrophysiological and cyclic AMP responses to beta-adrenergic receptor stimulation and catecholamine levels in cat and rabbit sympathetic ganglion.
1976
1976
Basic ethers of cyclohexylphenols with beta-blocking activity: synthesis and pharmacological study of exaprolol.
The paper describes the preparation and study of the pharmacological properties of a series of derivatives with the general… 
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