Skip to search formSkip to main contentSkip to account menu

RU 5135

Known as: 17-Azaandrost-16-en-11-one, 16-amino-3-hydroxy-, (3alpha,5beta)-, R 5135, RU-5135 
National Institutes of Health

Related topics

Related topics

3 relations

Broader (3)

AndrostanesAzasteroidsGABA Antagonists

Papers overview

Semantic Scholar uses AI to extract papers important to this topic.
1996
1996
The effect of GABA stimulation on GABAA receptor subunit protein and mRNA expression in rat cultured cerebellar granule cells
1 After 8 days in vitro, rat cerebellar granule cells were exposed to 1 mM γ‐aminobutyric acid (GABA) for periods of 1, 2, 4, 6… 
1992
1992
Glycinergic ligands modulate the rate of phosphorylation of the glycine receptor by protein kinase C.
1992
1992
Epileptogenic activity in the amygdala is not affected by the amidine steroid, R 5135
Highly Cited
1991
Highly Cited
1991
Agonist‐Dependent Internalization of γ‐Aminobutyric AcidA/Benzodiazepine Receptors in Chick Cortical Neurons
An impermeant benzodiazepine receptor ligand was prepared by derivatization of the aminobenzodiazepine 1012‐S with 4… 
1989
1989
Thermodynamics of Agonist and Antagonist Interaction with the Strychnine‐Sensitive Glycine Receptor
Abstract: The thermodynamic parameters associated with the interactions of agonists and antagonists with glycine receptors in rat… 
Highly Cited
1986
Highly Cited
1986
Kinetic regulation of convulsant (TBPS) binding by GABAergic agents.
The kinetics of specific [35S]-t-butylbicyclophosphorothionate (TBPS) binding was studied in rat brain synaptosomal membrane… 
Highly Cited
1985
Highly Cited
1985
Inhibitory influence of GABA on central serotonergic transmission. Raphe´nuclei as the neuroanatomical site of the GABAergic inhibition of cerebral serotonergic neurons
1985
1985
Glycine antagonism by RU 5135.
Highly Cited
1984
Highly Cited
1984
Convulsant potencies of tetrazoles are highly correlated with actions on GABA/benzodiazepine/picrotoxin receptor complexes in brain.
Highly Cited
1981
Highly Cited
1981
A steroid derivative, R 5135, antagonizes the GABA/benzodiazepine receptor interaction
By clicking accept or continuing to use the site, you agree to the terms outlined in our Privacy Policy (opens in a new tab), Terms of Service (opens in a new tab), and Dataset License (opens in a new tab)