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RU 5135
Known as:
17-Azaandrost-16-en-11-one, 16-amino-3-hydroxy-, (3alpha,5beta)-
, R 5135
, RU-5135
National Institutes of Health
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Related topics
Related topics
3 relations
Broader (3)
Androstanes
Azasteroids
GABA Antagonists
Papers overview
Semantic Scholar uses AI to extract papers important to this topic.
1996
1996
The effect of GABA stimulation on GABAA receptor subunit protein and mRNA expression in rat cultured cerebellar granule cells
K. Piatt
,
Raymond E. Zwartjes
,
D. Bristow
British Journal of Pharmacology
1996
Corpus ID: 40733348
1 After 8 days in vitro, rat cerebellar granule cells were exposed to 1 mM γ‐aminobutyric acid (GABA) for periods of 1, 2, 4, 6…
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1992
1992
Glycinergic ligands modulate the rate of phosphorylation of the glycine receptor by protein kinase C.
M. Vaello
,
A. Ruiz-Gómez
,
F. Mayor
Biochemical and Biophysical Research…
1992
Corpus ID: 25976579
1992
1992
Epileptogenic activity in the amygdala is not affected by the amidine steroid, R 5135
O. Kofman
,
R. Tarrasch
,
M. Mintz
,
Myslobodsky M.S.
Brain Research Bulletin
1992
Corpus ID: 4722677
Highly Cited
1991
Highly Cited
1991
Agonist‐Dependent Internalization of γ‐Aminobutyric AcidA/Benzodiazepine Receptors in Chick Cortical Neurons
M. Tehrani
,
E. M. Barnes
Journal of Neurochemistry
1991
Corpus ID: 22647104
An impermeant benzodiazepine receptor ligand was prepared by derivatization of the aminobenzodiazepine 1012‐S with 4…
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1989
1989
Thermodynamics of Agonist and Antagonist Interaction with the Strychnine‐Sensitive Glycine Receptor
A. Ruiz-Gómez
,
M. Garcia-Calvo
,
J. Vázquez
,
J. Marvizón
,
F. Valdivieso
,
F. Mayor
Journal of Neurochemistry
1989
Corpus ID: 24580173
Abstract: The thermodynamic parameters associated with the interactions of agonists and antagonists with glycine receptors in rat…
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Highly Cited
1986
Highly Cited
1986
Kinetic regulation of convulsant (TBPS) binding by GABAergic agents.
G. Maksay
,
M. Simonyi
Molecular Pharmacology
1986
Corpus ID: 22033766
The kinetics of specific [35S]-t-butylbicyclophosphorothionate (TBPS) binding was studied in rat brain synaptosomal membrane…
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Highly Cited
1985
Highly Cited
1985
Inhibitory influence of GABA on central serotonergic transmission. Raphe´nuclei as the neuroanatomical site of the GABAergic inhibition of cerebral serotonergic neurons
T. Nishikawa
,
B. Scatton
Brain Research
1985
Corpus ID: 35529638
1985
1985
Glycine antagonism by RU 5135.
D. R. Curtis
,
R. Malik
European Journal of Pharmacology
1985
Corpus ID: 33461987
Highly Cited
1984
Highly Cited
1984
Convulsant potencies of tetrazoles are highly correlated with actions on GABA/benzodiazepine/picrotoxin receptor complexes in brain.
R. Squires
,
E. Saederup
,
J. Crawley
,
P. Skolnick
,
S. Paul
Life Science
1984
Corpus ID: 22820289
Highly Cited
1981
Highly Cited
1981
A steroid derivative, R 5135, antagonizes the GABA/benzodiazepine receptor interaction
P. Hunt
,
S. Clements-Jewery
Neuropharmacology
1981
Corpus ID: 40422099
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