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Pteridinones

Pteridines with a 4-keto OXYGEN.
National Institutes of Health

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Pteridines

Papers overview

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2020
2020
Substituted pteridinones as p90 ribosomal S6 protein kinase (RSK) inhibitors: A structure-activity study.
The activity of p90 ribosomal S6 kinase 2 (RSK2) has emerged as an attractive target for cancer therapy due to its role in the… 
2020
2020
Molecular docking of substituted pteridinones and pyrimidines to the ATP-binding site of the N-terminal domain of RSK2 and associated MM/GBSA and molecular field datasets
The data have been obtained for a series of substituted pteridinones and pyrimidines that were developed based on BI-D1870 to… 
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2018
2018
Transition-Metal-Free С–С Coupling of 5,7-Dihydroxybenzopyrones with Quinoxalones and Pteridinones
A new synthetic protocol for nucleophilic substitution of hydrogen­ in quinoxalones and pteridinones by the action of 5,7-di… 
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2010
2010
4-methylpteridinones as orally active and selective PI3K/mTOR dual inhibitors.
Pteridinones were designed based on a non-selective kinase template. Because of the uniqueness of the PI3K and mTOR binding… 
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2005
2005
Pteridinones utilisees en tant qu'inhibiteurs des plk (polo-like-kinases)
L'invention concerne des composes de formule generale (I), dans laquelle L, Q1, Q2, X, Y, Ra, Rb, Rc, R1, R2, R3 et R4 sont tels… 
1993
1993
The synthesis of fluorine-containing pterins.
The introduction of fluorine into molecules has been well demonstrated to modify the biological properties significantly1. In… 
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