GR 113808

Known as: 1H-Indole-3-carboxylic acid, 1-methyl-, (1-(2-((methylsulfonyl)amino)ethyl)-4-piperidinyl)methyl ester, GR-113808, GR113808 
 
National Institutes of Health

Topic mentions per year

Topic mentions per year

1993-2017
051019932017

Papers overview

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2012
2012
BACKGROUND & AIMS 5-hydroxytryptamine receptor (5-HT(4)R) agonists promote gastrointestinal motility and attenuate visceral pain… (More)
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2007
2007
G protein-coupled receptors (GPCRs) signal through a limited number of G-protein pathways and play crucial roles in many… (More)
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2005
2005
Extracellular single-unit recordings in mouse brain slices were used to determine the effect of exogenously applied 5-HT on STN… (More)
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2003
2003
A large body of evidence supports a major role for the serotonin 5-HT(4) receptor in learning and memory and it is suggested that… (More)
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2000
2000
The present study was designed to investigate which subtypes of spinal 5-HT receptors are involved in 5-HT-induced… (More)
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1998
1998
1 5-Hydroxytryptamine (5-HT; 1 nM - 100 microM) concentration-dependently inhibited the amplitude and frequency of spontaneous… (More)
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1995
1995
GR-113808, a potent and selective 5-HT4 receptor antagonist, was infused through a microdialysis probe into the striatum and… (More)
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1994
1994
1. The 5-HT4 receptor has only recently been identified but has yet to be cloned. This paper describes the pharmacology of a… (More)
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1993
1993
1. The mode of antagonism of 5-hydroxytryptamine (5-HT)-induced positive inotropic effects by the highly selective 5-HT4 receptor… (More)
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1993
1993
1. The 5-HT4 receptor antagonist, GR113808, has been radiolabelled to a high specific activity with tritium. 2. Characterization… (More)
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