G-protein coupled receptor kinase activity

Known as: G protein coupled receptor phosphorylating protein kinase activity, GPCR kinase activity, ATP:G-protein-coupled receptor phosphotransferase activity 
Catalysis of the reaction: ATP + G-protein coupled receptor = ADP + G-protein coupled receptor phosphate. [GOC:dph]
National Institutes of Health

Topic mentions per year

Topic mentions per year

1993-2017
051019932017

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2012
2012
Seven-transmembrane receptors (7TMRs) are involved in nearly all aspects of chemical communications and represent major drug… (More)
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2011
2011
AIMS prolonged P2Y-receptor signalling can cause vasoconstriction leading to hypertension, vascular smooth muscle hypertrophy… (More)
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2009
2009
During conditions of moderate sodium excess, the dopaminergic system regulates blood pressure and water and electrolyte balance… (More)
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2005
2005
The H1 histamine receptor (H1HR) is a member of the G protein-coupled receptor superfamily and regulates numerous cellular… (More)
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2002
2002
BACKGROUND The D1 dopamine receptor, expressed in several nephron segments, participates in the regulation of water and… (More)
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2000
2000
G-protein-coupled receptor kinases (GRKs) are involved in the regulation of many G-protein-coupled receptors. As opposed to the… (More)
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1998
1998
The G protein-coupled receptor kinase GRK6 undergoes posttranslational modification by palmitoylation. Palmitoylated GRK6 is… (More)
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1997
1997
G protein-coupled receptor kinases (GRKs) specifically recognize and phosphorylate the hormone-occupied form of numerous G… (More)
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Highly Cited
1997
Highly Cited
1997
Although endothelin-1 can elicit prolonged physiologic responses, accumulating evidence suggests that rapid desensitization… (More)
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1994
1994
G protein-coupled receptor kinases (GRKs) play an important role in mediating agonist-specific desensitization of numerous G… (More)
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