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CI 966
Known as:
CI-966
National Institutes of Health
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Related topics
Related topics
1 relation
Broader (1)
Pyridines
Papers overview
Semantic Scholar uses AI to extract papers important to this topic.
2019
2019
GRID-independent molecular descriptor analysis and molecular docking studies to mimic the binding hypothesis of γ-aminobutyric acid transporter 1 (GAT1) inhibitors
Sadia Zafar
,
Ishrat Jabeen
PeerJ
2019
Corpus ID: 59605434
Background The γ-aminobutyric acid (GABA) transporter GAT1 is involved in GABA transport across the biological membrane in and…
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Highly Cited
2005
Highly Cited
2005
First Demonstration of a Functional Role for Central Nervous System Betaine/γ-Aminobutyric Acid Transporter (mGAT2) Based on Synergistic Anticonvulsant Action among Inhibitors of mGAT1 and mGAT2
H. White
,
W. P. Watson
,
+11 authors
A. Schousboe
Journal of Pharmacology and Experimental…
2005
Corpus ID: 30717285
In a recent study, EF1502 [N-[4,4-bis(3-methyl-2-thienyl)-3-butenyl]-3-hydroxy-4-(methylamino)-4,5,6,7-tetrahydrobenzo [d…
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2001
2001
Synthesis of novel gamma-aminobutyric acid (GABA) uptake inhibitors. 5.(1) Preparation and structure-activity studies of tricyclic analogues of known GABA uptake inhibitors.
K. Andersen
,
J. Sorensen
,
+5 authors
Michael D B Swedberg
Journal of Medicinal Chemistry
2001
Corpus ID: 21334214
On the basis of the SAR of a series of known gamma-aminobutyric acid (GABA) uptake inhibitors, including 4 (SKF 89976), new…
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Review
2000
Review
2000
GABA potentiation: a logical pharmacological approach for the treatment of acute ischaemic stroke
A. Green
,
A. Hainsworth
,
D. Jackson
Neuropharmacology
2000
Corpus ID: 39073036
Highly Cited
1997
Highly Cited
1997
Characterization of the anticonvulsant properties of Ganaxolone (CCD 1042; 3α-hydroxy-3β-methyl-5α-pregnan-20-one), a selective, high-affinity, steroid modulator of the γ-aminobutyric acid(A…
R. B. Carter
,
P. Wood
,
+10 authors
K. Gee
1997
Corpus ID: 10518047
Ganaxolone (CCD 1042) is a 3b-methyl-substituted analog of the endogenous neuroactive steroid 3a-hydroxy-5a-pregnan20-one…
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1995
1995
CI-966, a GABA uptake inhibitor, antagonizes ischemia-induced neuronal degeneration in the gerbil.
J. Phillis
General Pharmacology
1995
Corpus ID: 33929585
Highly Cited
1994
Highly Cited
1994
Tiagabine, SK&F 89976-A, CI-966, and NNC-711 are selective for the cloned GABA transporter GAT-1.
L. Borden
,
T. G. Murali Dhar
,
K. E. Smith
,
R. Weinshank
,
T. Branchek
,
C. Gluchowski
European Journal of Pharmacology
1994
Corpus ID: 38242528
1994
1994
Discriminative stimulus effects of presynaptic GABA agonists in pentobarbital-trained rats
D. M. Grech
,
R. Balster
Pharmacology, Biochemistry and Behavior
1994
Corpus ID: 8783707
1993
1993
Identification of a pyridinium metabolite in human urine following a single oral dose of 1-[2-[bis[4-(trifluoromethyl)phenyl]methoxy]ethyl]- 1,2,5,6-tetrahydro-3-pyridinecarboxylic acid…
L. Radulovic
,
T. Woolf
,
+4 authors
T. Chang
Chemical Research in Toxicology
1993
Corpus ID: 434726
Single-dose administration of 50 mg of 1-[2-[bis[4- (trifluoromethyl)phenyl]methoxy]ethyl]-1,2,5,6-tetrahydro-3…
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1990
1990
Systemic CI-966, a new gamma-aminobutyric acid uptake blocker, enhances gamma-aminobutyric acid action in CA1 pyramidal layer in situ.
U. Ebert
,
K. Krnjević
Canadian Journal of Physiology and Pharmacology
1990
Corpus ID: 25466934
A new potent, blood-brain barrier permeable gamma-aminobutyric acid (GABA) uptake blocker, 1-[2-[bis[4-(trifluoromethyl)-phenyl…
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