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CGP 12177

Known as: 2H-Benzimidazol-2-one, 4-(3-((1,1-dimethylethyl)amino)-2-hydroxypropoxy)-, CGP-12177 
National Institutes of Health

Related topics

Related topics

4 relations

Broader (3)

Adrenergic beta-AgonistsAdrenergic beta-AntagonistsPropanolamines

Narrower (1)

CGP 12177A

Papers overview

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2017
2017
Gherbi, Karolina and May, Lauren T. and Baker, Jillian G. and Briddon, Stephen J. and Hill, Stephen J. (2015) Negative cooperativity across 1-adrenoceptor homodimers provides insights into the nature…
At the b1-adrenoceptor, CGP 12177 potently antagonizes agonist responses at the primary highaffinity catecholamine conformation… 
1989
1989
Microwave attenuation of ethanol-induced interactions with noradrenergic neurotransmitter systems.
Research suggests that microwave (MW) irradiation can attenuate ethanol (EtOH)-induced hypothermia in a manner that may depend… 
Highly Cited
1986
Highly Cited
1986
In vivo regulation of beta-adrenergic receptors on human mononuclear leukocytes: assessment of receptor number, location, and function after posture change, exercise, and isoproterenol infusion.
We studied the regulation of beta-adrenergic receptors in human mononuclear leukocytes (MNL). Total receptor number was… 
1986
1986
Desensitization and redistribution of beta-adrenergic receptors on human mononuclear leukocytes.
We have used intact human mononuclear leukocytes (MNL) to examine desensitization of beta-adrenergic receptors in normal… 
1984
1984
Some unique properties of CGP-12177.
CGP-12177, like isoproterenol, has a lower affinity for desensitized receptors. Experiments were performed to study whether this… 
1984
1984
Desensitized beta-adrenoceptors of C6-glioma cells have distinct binding properties
SummaryWhen C6-rat glioma cells were incubated for 20 min with beta-adrenoceptor agonists, a part of the beta-adrenoceptors was… 
1984
1984
Recovery of beta-adrenoceptors and cyclic AMP response after long term treatment of intact heart cells with beta-blockers.
We have studied the recovery of receptor binding and of isoprenaline-stimulated cyclic AMP responses after chronic (2-5 days… 
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