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4-methylcoumarin 7-O-sulfamate

Known as: COUMATE 
National Institutes of Health

Related topics

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2 relations

Broader (2)

CoumarinsSulfonamides

Papers overview

Semantic Scholar uses AI to extract papers important to this topic.
2019
2019
Synthesis and evaluation of coumate analogues as estrogen receptor inhibitors for breast cancer therapy
A sulphatase inhibitor 667 COUMATE is in clinical trials for estrogen-positive breast cancer therapy for postmenopausal women… 
2014
2014
Steroid sulfatase mediated growth Sof human MG-63 pre-osteoblastic cells
Review
2013
Review
2013
Steroid sulfatase inhibitors: promising new therapy for breast cancer.
  • H. Sadozai
  • JPMA. The Journal of the Pakistan Medical…
  • 2013
  • Corpus ID: 163269
Manipulation of the hormone oestrogen has been used for decades to treat hormone-dependent breast cancer. Currently, aromatase… 
Review
2008
Review
2008
Recent developments of steroid sulfatase inhibitors as anti-cancer agents.
The steroid sulfatase (STS) enzyme plays a pivotal role in the formation of biologically active steroid hormones. Its involvement… 
2005
2005
Inhibition of steroid sulfatase by 667 COUMATE (STX64): a new treatment paradigm for breast cancer
2004
2004
The role of steroid sulphatase in regulating the oestrogenicity of oestrogen sulphamates.
2004
2004
La stéroi͏̈de sulfatase : localisation cérébrale lors du développement postnatal : détermination cellulaire de son expression : implications comportementales liées à son inhibition par le COUMATE
La steroide sulfatase (STS) est une enzyme essentielle dans le metabolisme des neurosteroides. Elle permet le controle du rapport… 
2003
2003
Development of a sensitive high-performance liquid chromatography method for the detection of 667 COUMATE in vivo
2002
2002
The design, synthesis, and biochemical evaluation of derivatives of biphenyl sulfamate-based compounds as novel inhibitors of estrone sulfatase.
2002
2002
Inhibition of estrone sulfatase (ES) by derivatives of 4-[(aminosulfonyl)oxy] benzoic acid.
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