Synthesis of 2-aryl-oxazolo[4,5-c]quinoline-4(5H)-ones and 2-aryl-thiazolo[4,5-c]quinoline-4(5H)-ones.

@article{Hodgetts2003SynthesisO2,
  title={Synthesis of 2-aryl-oxazolo[4,5-c]quinoline-4(5H)-ones and 2-aryl-thiazolo[4,5-c]quinoline-4(5H)-ones.},
  author={K. Hodgetts and Mark T. Kershaw},
  journal={Organic letters},
  year={2003},
  volume={5 16},
  pages={
          2911-4
        }
}
  • K. Hodgetts, Mark T. Kershaw
  • Published 2003
  • Chemistry, Medicine
  • Organic letters
    • [reaction: see text] Novel and highly efficient syntheses of oxazolo[4,5-c]quinoline-4(5H)-ones (1) and thiazolo[4,5-c]quinoline-4(5H)-ones (2) from ethyl 2-chlorooxazole-4-carboxylate (4) and ethyl 2-bromo-5-chlorothiazole-4-carboxylate (13), respectively, are described. 
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