Synthesis of 10-Acetyl-5,8-dideazafolic Acid (I): A Potent Inhibitor of Glycinamide Ribonucleotide Transformylase.

@article{Caperelli1987SynthesisO1,
  title={Synthesis of 10-Acetyl-5,8-dideazafolic Acid (I): A Potent Inhibitor of Glycinamide Ribonucleotide Transformylase.},
  author={Carol A. Caperelli and James P. Conigliaro},
  journal={ChemInform},
  year={1987},
  volume={18}
}
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References

Synthesis of 10-acetyl-5,8-dideazafolic acid: a potent inhibitor of glycinamide ribonucleotide transformylase.
TLDR
This quinazoline folate analogue showed no activity as a substrate for the folate-requiring de novo purine biosynthetic enzyme glycinamide ribonucleotide transformylase isolated from the murine lymphoma cell line L5178Y, but proved to be a potent competitive inhibitor.