Synthesis and collagenase inhibition of new glycosides of aranciamycinone: the aglycon of the naturally occurring antibiotic aranciamycin.

@article{Bols1992SynthesisAC,
  title={Synthesis and collagenase inhibition of new glycosides of aranciamycinone: the aglycon of the naturally occurring antibiotic aranciamycin.},
  author={M. Bols and L. Binderup and J. Hansen and P. Rasmussen},
  journal={Carbohydrate research},
  year={1992},
  volume={235},
  pages={
          141-9
        }
}
  • M. Bols, L. Binderup, +1 author P. Rasmussen
  • Published 1992
  • Chemistry, Medicine
  • Carbohydrate research
  • Glycosides of aranciamycinone were prepared by glycosylation with sugar acetates and trimethylsilyl triflate in dichloromethane. Glycosides of the following sugars were prepared: alpha-L-rhamnopyranose, beta-D-glucopyranose, beta-D-ribopyranose, beta-D-xylopyranose, alpha-L-fucopyranose, 2-azido-2,6-dideoxy-alpha-L-mannopyranose, 2,6-dideoxy-alpha-L-arabino-hexopyranose, 3,6-dideoxy-alpha-L-arabino-hexopyranose, and 4,6-dideoxy-alpha-L-lyxo-hexopyranose. The new glycosides were tested for… CONTINUE READING
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