Studies on the structure-activity relationship of bicifadine analogs as monoamine transporter inhibitors.

Abstract

Compounds with various activities and selectivities were discovered through structure-activity relationship studies of bicifadine analogs as monoamine transporter inhibitors. The norepinephrine-selective 2-thienyl compound S-6j was efficacious in a rodent pain model. 
DOI: 10.1016/j.bmcl.2008.05.077

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