Scope of the palladium-catalyzed aryl borylation utilizing bis-boronic acid.

Abstract

The Suzuki-Miyaura reaction has become one of the more useful tools for synthetic organic chemists. Until recently, there did not exist a direct way to make the most important component in the coupling reaction, namely the boronic acid. Current methods to make boronic acids often employ harsh or wasteful reagents to prepare boronic acid derivatives and… (More)
DOI: 10.1021/ja303181m

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10 Figures and Tables