Role of GABAB receptors in GABA and baclofen-induced inhibition of adult rat cerebellar interpositus nucleus neurons in vitro
@article{Chen2005RoleOG, title={Role of GABAB receptors in GABA and baclofen-induced inhibition of adult rat cerebellar interpositus nucleus neurons in vitro}, author={Kun Chen and Hong-Zhao Li and Na Ye and Jun Zhang and Jian-jun Wang}, journal={Brain Research Bulletin}, year={2005}, volume={67}, pages={310-318} }
38 Citations
Orexins Excite Neurons of the Rat Cerebellar Nucleus Interpositus Via Orexin 2 Receptors In Vitro
- Biology, PsychologyThe Cerebellum
- 2009
It is demonstrated that orexins excite the cerebellar IN neurons through OX2R and suggest that the central orexinergic nervous system may actively participate in motor control through its modulation on one of the final outputs of the spinocerebellum.
A REVIEW ON GAMMA-AMINOBUTYRIC ACID (GABA) AND ITS RECEPTORS
- Biology
- 2012
The pharmacology of these novel subtypes of GABA receptors are expected to mediate the lateral inhibition of light responses and have been shown to inhibit transmitter release at bipolar cell terminals and may yield important therapeutic agents.
Contradictory effects of GABA-B receptor agonists on cortical epileptic afterdischarges in immature rats
- Biology, PsychologyBrain Research Bulletin
- 2008
Intrathecal baclofen, a GABAB receptor agonist, inhibits the expression of p-CREB and NR2B in the spinal dorsal horn in rats with diabetic neuropathic pain.
- BiologyCanadian journal of physiology and pharmacology
- 2014
Activation of GABAB receptor by baclofen attenuates diabetic neuropathic pain, which may partly be accomplished via down-regulating the expression of p-CREB and NR2B.
The Role of GABA Receptor Agonists in Anesthesia and Sedation
- BiologyCNS Drugs
- 2017
An overview of the role that GABAAR agonists currently play in sedation and anesthesia is provided, in addition to discussing the future role of novel GABAar agonists in anesthesia and sedation.
Histamine improves rat rota-rod and balance beam performances through H2 receptors in the cerebellar interpositus nucleus
- BiologyNeuroscience
- 2006
Effects of GABAB receptor antagonists CGP63360, CGP76290A and CGP76291A on learning and memory processes in rodents
- Biology, Psychology
- 2007
It may be concluded that the obtained results on the GABAB receptor antagonists could contribute to their pharmacological characteristics and might be of interest for potential clinical implication.
A Substituted Anilino Enaminone Acts as a Novel Positive Allosteric Modulator of GABAA Receptors in the Mouse Brain
- Biology, ChemistryJournal of Pharmacology and Experimental Therapeutics
- 2011
Clinical use of anilino enaminones as anticonvulsants in seizures and as a potential anxiolytic in mental disorders are suggested.
Allosteric Modulation of GABAA Receptors by an Anilino Enaminone in an Olfactory Center of the Mouse Brain
- BiologyPharmaceuticals
- 2014
This anilino enaminone KRS-5Me-4-OCF3 emerges as a candidate for clinical use as an anticonvulsant agent in the battle against epileptic seizures.
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