Regulation of central 5-HT2A receptors: a review of in vivo studies

@article{Eison1995RegulationOC,
  title={Regulation of central 5-HT2A receptors: a review of in vivo studies},
  author={A. S. Eison and U. L. Mullins},
  journal={Behavioural Brain Research},
  year={1995},
  volume={73},
  pages={177-181}
}
Numerous investigations have studied in vivo regulation of central 5-HT2A receptors. The majority of pharmacological studies point to non-classical regulation of this site. Serotonergic denervation does not modify 5-HT2A receptor density or second messenger responses (phosphoinositide hydrolysis). 5-HT2A receptor downregulation is produced by the chronic administration of 5-HT2A receptor agonists and uniquely among monoamine receptors by antagonists. Several classes of psychotherapeutic agents… Expand
Desensitization of 5-HT1A Receptors by 5-HT2A Receptors in Neuroendocrine Neurons in Vivo
Selective and divergent regulation of cortical 5-HT(2A) receptors in rabbit.
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