Reevaluating the synthesis of 2,5‐disubstituted‐1 H ‐benzimidazole derivatives by different green activation techniques and their biological activity as antifungal and antimicrobial inhibitor

@article{PenieresCarrillo2019ReevaluatingTS,
  title={Reevaluating the synthesis of 2,5‐disubstituted‐1
 H
 ‐benzimidazole derivatives by different green activation techniques and their biological activity as antifungal and antimicrobial inhibitor},
  author={Jos{\'e} Guillermo Penieres-Carrillo and Hulme R{\'i}os-Guerra and Javier P{\'e}rez-Flores and Braulio Rodr{\'i}guez‐Molina and {\'A}ngeles Torres-Reyes and Francisco Barrera-T{\'e}llez and Jessica V. Gonz{\'a}lez-Carrillo and Lessly Moreno‐Gonz{\'a}lez and Alejandro Mart{\'i}nez-Z{\'a}ldivar and Juan‐Jes{\'u}s Nolasco‐Fidencio and Audif{\'a}s-Salvador Matus-Meza and Ricardo Alfredo Luna-Mora},
  journal={Journal of Heterocyclic Chemistry},
  year={2019},
  volume={57},
  pages={436-455}
}
2 Citations
Solid-state zwitterionic tautomerization of 2-((5-methyl-1H-pyrazol-3-yl)methyl)-1H-benzimidazole: Synthesis, characterization, DFT calculation and docking studies
Abstract The synthesis, characterization and single crystal X-Ray diffraction structure of 2-((5-methyl-1H-pyrazol-3-yl)methyl)-1H-benzimidazole are reported. The physicochemical characterization ofExpand
Synthesis, bioevaluation and docking studies of some 2-phenyl-1H-benzimidazole derivatives as anthelminthic agents against the nematode Teladorsagia circumcincta.
TLDR
Docking studies of most potent compounds in a modelled Teladorsagia tubulin indicated an inverted orientation for BZ 1 in the colchicine binding site, probably due to its fair interaction with glutamic acid at codon 198, which could justify its inactivity against the resistant strain of T. circumcincta. Expand

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