Receptor interaction profiles of novel psychoactive tryptamines compared with classic hallucinogens.

@article{Rickli2016ReceptorIP,
  title={Receptor interaction profiles of novel psychoactive tryptamines compared with classic hallucinogens.},
  author={Anna Rickli and Olivier D Moning and Marius C. Hoener and Matthias E Liechti},
  journal={European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology},
  year={2016},
  volume={26 8},
  pages={1327-37}
}
The present study investigated interactions between the novel psychoactive tryptamines DiPT, 4-OH-DiPT, 4-OH-MET, 5-MeO-AMT, and 5-MeO-MiPT at monoamine receptors and transporters compared with the classic hallucinogens lysergic acid diethylamide (LSD), psilocin, N,N-dimethyltryptamine (DMT), and mescaline. We investigated binding affinities at human monoamine receptors and determined functional serotonin (5-hydroxytryptamine [5-HT]) 5-HT2A and 5-HT2B receptor activation. Binding at and the… CONTINUE READING
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