Potency of progestogens used in hormonal therapy: Toward understanding differential actions

@article{Hapgood2014PotencyOP,
  title={Potency of progestogens used in hormonal therapy: Toward understanding differential actions},
  author={Janet P. Hapgood and Donita Africander and Renate Louw and Ramesh M. Ray and Julia Rohwer},
  journal={The Journal of Steroid Biochemistry and Molecular Biology},
  year={2014},
  volume={142},
  pages={39-47}
}

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Differential Glucocorticoid Receptor‐Mediated Effects on Immunomodulatory Gene Expression by Progestin Contraceptives: Implications for HIV‐1 Pathogenesis

It is reported that MPA, unlike NET and progesterone, represses inflammatory genes in human PBMCs in a dose‐dependent manner, via the glucocorticoid receptor (GR), at concentrations within the physiologically relevant range.

Recent advances in structure of progestins and their binding to progesterone receptors

The aim of this review is to describe the basic structure of PR agonists and antagonists as well as the recent treatments for illness associated with the progesterone receptor.
...

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