Pharmacological profile of mephedrone analogs and related new psychoactive substances

@article{Luethi2018PharmacologicalPO,
  title={Pharmacological profile of mephedrone analogs and related new psychoactive substances},
  author={D. Luethi and Karolina E. Kolaczynska and Luca Docci and S. Kr{\"a}henb{\"u}hl and M. Hoener and M. Liechti},
  journal={Neuropharmacology},
  year={2018},
  volume={134},
  pages={4-12}
}
BACKGROUND Mephedrone is a synthetic cathinone and one of the most popular recreationally used new psychoactive substances. The aim of the present study was to characterize the in vitro pharmacology of novel analogs of mephedrone and related newly emerged designer stimulants. METHODS We determined norepinephrine, dopamine, and serotonin transporter inhibition potencies and monoamine release in transporter-transfected human embryonic kidney 293 cells. We also assessed monoamine receptor and… Expand
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  • D. Luethi, M. Liechti
  • Chemistry, Medicine
  • The international journal of neuropsychopharmacology
  • 2018
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