Partial agonist activity of carteolol on atypical beta-adrenoceptors in the guinea pig duodenum.
@article{Horinouchi2000PartialAA, title={Partial agonist activity of carteolol on atypical beta-adrenoceptors in the guinea pig duodenum.}, author={Takahiro Horinouchi and Katsuo Koike}, journal={European journal of pharmacology}, year={2000}, volume={403 1-2}, pages={ 133-8 } }
6 Citations
Agonistic activity of SR59230A at atypical beta-adrenoceptors in guinea pig gastric fundus and duodenum.
- Biology, MedicineEuropean journal of pharmacology
- 2001
Partial agonistic activity of labetalol, the arylethanolamine, on beta 3-adrenoceptors in the guinea-pig gastric fundus.
- Biology, ChemistryAutonomic & autacoid pharmacology
- 2002
The results indicate that labetalol, the arylethanolamine, acts as a partial agonist on beta3-adrenoceptors in the guinea-pig gastric fundus.
Further evidence that (+/-)-carteolol-induced relaxation is mediated by beta2-adrenoceptors but not by beta3-adrenoceptors in the guinea pig taenia caecum.
- BiologyJournal of smooth muscle research = Nihon Heikatsukin Gakkai kikanshi
- 2000
The results suggest that the relaxant effects of (+/-)-carteolol in the guinea pig taenia caecum are mediated by beta2-adrenoceptors but not by beta3- adrenOceptors.
Further characterization of β3-adrenoceptors in the guinea pig gastric fundus: stereoselectivity, β-adrenoceptor alkylation, and structure-activity relationship
- Chemistry, Biology
- 2001
Isomeric activity ratios for isomers of isoprenaline and noradrenaline were less than those obtained for activation of β1- and β2-adrenoceptors in the guinea pig atria and trachea, respectively.
β2-Adrenoceptor-mediated intrinsic sympathomimetic activity of carteolol: an in vivo study
- Biology, MedicineNaunyn-Schmiedeberg's Archives of Pharmacology
- 2004
The fact that the cardiovascular effects of carteolol were not attenuated by the β1-adrenoceptor blocker bisoprolol and, on the other, carteoolol significantly decreased lymphocyte β2-adRenoceptor density and function is in favour of the idea that the ISA of cartaolol is mediated byβ2- adrenoceptors.
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