One-step conversion of azine N-oxides to alpha-1,2,4-triazolo-, 1,2,3-triazolo, imidazolo-, and pyrazoloheteroarenes.

  • John M Keith
  • Published 2010 in The Journal of organic chemistry

Abstract

Pyridine, quinoline, isoquinoline, azaindole, and pyrimidine N-oxides were converted to their alpha-triazole and alpha-diazole derivatives by treatment with the corresponding p-toluenesulfonylazoles and Hunig's base at elevated temperatures.

DOI: 10.1021/jo1001017

Cite this paper

@article{Keith2010OnestepCO, title={One-step conversion of azine N-oxides to alpha-1,2,4-triazolo-, 1,2,3-triazolo, imidazolo-, and pyrazoloheteroarenes.}, author={John M Keith}, journal={The Journal of organic chemistry}, year={2010}, volume={75 8}, pages={2722-5} }