One-Pot Tandem Synthesis of 2-Arylquinazolines by a Multicomponent Cyclization Reaction

@inproceedings{Ye2013OnePotTS,
  title={One-Pot Tandem Synthesis of 2-Arylquinazolines by a Multicomponent Cyclization Reaction},
  author={Leping Ye and L Yu and Lijun Zhu and Xiaodong Xia},
  booktitle={Molecules},
  year={2013}
}
A series of 2-arylquinazolines have been synthesized in moderate to excellent yields by one-pot tandem reaction of (2-aminophenyl)methanols, aldehydes and ceric ammonium nitrate (CAN). The utility of this transformation was demonstrated by its compatibility with a wide range of functional groups. Thus, the method represents a simple and practical procedure to access 2-arylquinazolines. 

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