Novel solid-phase synthesis of 1,5-benzothiazepine-4-one derivatives

@inproceedings{Morton2000NovelSS,
  title={Novel solid-phase synthesis of 1,5-benzothiazepine-4-one derivatives},
  author={George C. Morton and Joseph M. Salvino and Richard F. Labaudini{\`e}re and Timothy F. Herpin},
  year={2000}
}
Abstract A new solid-phase efficient route to 1,5-benzothiazepine-4-one derivatives is reported. The synthesis exploits the variety of halo-nitrobenzene derivatives available and the facile substitution of the benzamide nitrogen. A wide range of derivatives can be obtained in excellent purity.