Iodinated photoreactive vasopressin antagonists: labelling of hepatic vasopressin receptor subunits.

Abstract

To identify and characterize V1 vasopressin receptors, photoreactive antagonists of the glycogenolytic and vasoconstrictor activity of vasopressin have been synthesized. The following analogues with 3-mercapto-3,3-cyclopentamethylene-propionic acid (Mca) and N-methylalanine (MeAla) in position 1 and 7 of vasopressin (VP) were effective V1 antagonists: [Mca1… (More)

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Cite this paper

@article{Fahrenholz1986IodinatedPV, title={Iodinated photoreactive vasopressin antagonists: labelling of hepatic vasopressin receptor subunits.}, author={Falk Fahrenholz and Elzbieta Kojro and M. Mueller and Rob Boer and Raymond C. Loehr and Zbigniew Grzonka}, journal={European journal of biochemistry}, year={1986}, volume={161 2}, pages={321-8} }