In vivo estrogen bioactivities and in vitro estrogen receptor binding and transcriptional activities of anticoagulant synthetic 17β-aminoestrogens

@article{Jaimez2000InVE,
  title={In vivo estrogen bioactivities and in vitro estrogen receptor binding and transcriptional activities of anticoagulant synthetic 17$\beta$-aminoestrogens},
  author={R. Jaimez and A. Cooney and K. Jackson and A. E. Lemus and F. Larrea},
  journal={The Journal of Steroid Biochemistry and Molecular Biology},
  year={2000},
  volume={73},
  pages={59-66}
}
Estrogenic activities of the two 17beta-aminoestrogen (AE) derivatives, prolame and butolame, were studied upon coagulation, serum luteinizing hormone (LH) and uterine weight, including endometrial morphology in castrated female rats. We have also investigated the ability of these two compounds, as well as another AE pentolame, to activate transcription through the estrogen receptor alpha (ERalpha) and the estrogen receptor beta (ERbeta). Administration of prolame and butolame to castrated… Expand
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