Identification of a Highly Potent and Selective DNA-Dependent Protein Kinase (DNA-PK) Inhibitor (NU7441) by Screening of Chromenone Libraries.

@article{Leahy2005IdentificationOA,
  title={Identification of a Highly Potent and Selective DNA-Dependent Protein Kinase (DNA-PK) Inhibitor (NU7441) by Screening of Chromenone Libraries.},
  author={Justin J. J. Leahy and Bernard T Golding and Roger John Griffin and Ian R Hardcastle and Caroline J. Richardson and Laurent Jean Martin Rigoreau and Graeme C M Smith},
  journal={ChemInform},
  year={2005},
  volume={36}
}
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References

Identification of a highly potent and selective DNA-dependent protein kinase (DNA-PK) inhibitor (NU7441) by screening of chromenone libraries.
A solution-phase multiple-parallel synthesis approach was employed for the preparation of 6-, 7- and 8-aryl-substituted chromenone libraries, which were screened as inhibitors of the DNA repairExpand