H1‐antihistamines: inverse agonism, anti‐inflammatory actions and cardiac effects

@article{Leurs2002H1antihistaminesIA,
  title={H1‐antihistamines: inverse agonism, anti‐inflammatory actions and cardiac effects},
  author={R. Leurs and M. Church and M. Taglialatela},
  journal={Clinical & Experimental Allergy},
  year={2002},
  volume={32}
}
  • R. Leurs, M. Church, M. Taglialatela
  • Published 2002
  • Chemistry, Medicine
  • Clinical & Experimental Allergy
  • This review addresses novel concepts of histamine H1‐receptor function and attempts to relate them to the anti‐inflammatory effects of H1‐antihistamines. Furthermore, the molecular mechanisms underlying the cardiotoxic effects of H1‐antihistamines are discussed. 
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