Generation of potent and selective kinase inhibitors by combinatorial biosynthesis of glycosylated indolocarbazoles.

@article{Snchez2009GenerationOP,
  title={Generation of potent and selective kinase inhibitors by combinatorial biosynthesis of glycosylated indolocarbazoles.},
  author={C. S{\'a}nchez and Aaroa P Salas and Alfredo F. Bra{\~n}a and Martina Palomino and Antonio Pineda-Lucena and Rodrigo J. Carbajo and Carmen M{\'e}ndez and Francisco Mor{\'i}s and Jos{\'e} A Salas},
  journal={Chemical communications},
  year={2009},
  volume={27},
  pages={4118-20}
}
We report the generation of novel glycosylated indolocarbazoles by combinatorial biosynthesis, and the identification of two novel potent and selective compounds inhibitors of JAK2 and Ikkb kinases. 

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