Evidence for various tryptamines and related compounds acting as substrates of the platelet 5-hydroxytryptamine transporter

@article{Wlfel2004EvidenceFV,
  title={Evidence for various tryptamines and related compounds acting as substrates of the platelet 5-hydroxytryptamine transporter},
  author={R. W{\"o}lfel and K. Graefe},
  journal={Naunyn-Schmiedeberg's Archives of Pharmacology},
  year={2004},
  volume={345},
  pages={129-136}
}
  • R. Wölfel, K. Graefe
  • Published 2004
  • Chemistry, Medicine
  • Naunyn-Schmiedeberg's Archives of Pharmacology
SummaryThe aim of the present study was to answer the question whether amines other than 5-hydroxytryptamine (5-HT) and tryptamine act as substrates of the platelet 5-HT transporter. To this end, a large number of tryptamines, 5-HT receptor agonists and phenethylamines (which had IC50 values for 3H-5-HT uptake inhibition of 145–24500 nmol l−1) was examined in rabbit platelets in order to determine their ability to induce an outward transport of 3H-5-HT Platelets (the MAO of which was blocked… Expand
The recreational tryptamine 5-MeO-DALT (N,N-diallyl-5-methoxytryptamine): A brief review
...
1
2
...

References

SHOWING 1-10 OF 35 REFERENCES
Effects of imipramine and some tryptamine derivatives on the efflux of 3H-5-hydroxytryptamine from rabbit platelets.
Neurochemical characterization of a new potent and selective serotonin uptake inhibitor: Lu 10-171
  • J. Hyttel
  • Chemistry, Medicine
  • Psychopharmacology
  • 2004
Comparison of the pharmacological characteristics of 5 HT1 and 5 HT2 binding sites with those of serotonin autoreceptors which modulate serotonin release
Uptake of 5-hydroxytryptamine by platelets.
  • R. S. Stacey
  • Medicine
  • British journal of pharmacology and chemotherapy
  • 1961
Mechanism of imipramine inhibition of platelet 5-hydroxytryptamine transport.
Citalopram — Pharmacological profile of a specific serotonin uptake inhibitor with antidepressant activity
  • J. Hyttel
  • Medicine, Chemistry
  • Progress in Neuro-Psychopharmacology and Biological Psychiatry
  • 1982
5‐HYDROXYTRYPTAMINE AND DOPAMINE TRANSPORT BY RAT AND HUMAN BLOOD PLATELETS
...
1
2
3
4
...