Evaluation of a new beta-adrenergic blocking agent, carteolol, based on metabolic responses in rats-II. Blockade by carteolol of the epinephrine-and isoproterenol-induced increases of tissue and blood cyclic AMP in vivo.

@article{Saitoh1976EvaluationOA,
  title={Evaluation of a new beta-adrenergic blocking agent, carteolol, based on metabolic responses in rats-II. Blockade by carteolol of the epinephrine-and isoproterenol-induced increases of tissue and blood cyclic AMP in vivo.},
  author={Yuichi Saitoh and Seiji Morita and Yasuo Irie and Hideaki Kohri},
  journal={Biochemical pharmacology},
  year={1976},
  volume={25 16},
  pages={
          1843-9
        }
}
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23 Citations

Effect of a selective β2-adrenoceptor agonist, procaterol, on tissue cyclic AMP level: Its determination after tissue fixation by microwave irradiation

Age-related changes of in vivo β-adrenergic responsiveness in normotensive and spontaneously hypertensive rats

Effects of cardiotoxic doses of adrenergic amines on myocardial cyclic AMP.

Evaluation of a new beta-adrenoceptor agonist, procaterol, based on metabolic responses in rats.

The plasma cyclic AMP response to catecholamines as potentiated by phentolamine in rats.

Increases in plasma cyclic AMP dependent on endogenous catecholamines.

Adrenomedullary and β-adrenergic participation in enhanced sympathetic pressor responses of spontaneously hypertensive rats

Plasma cyclic GMP: response to cholinergic agents.

  • M. HonmaM. Ui
  • Biology, Chemistry
    European journal of pharmacology
  • 1978

Plasma cyclic AMP in the morphine-tolerant rat.

The tissue content of cyclic AMP in rats after microwave irradiation in vivo.

It is concluded that rapid tissue fixation by microwave irradiation may provide a useful means for obtaining reliable values of the tissue cyclic AMP content.

References

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The results suggest that NE interacts with at least two types of receptors (analogous to alpha and beta ) whereas ISO appears to react with a single type (analagous to beta ).

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CHARACTERISTICS OF THE CATECHOLAMINE AND HISTAMINE RECEPTOR SITES MEDIATING ACCUMULATION OF CYCLIC ADENOSINE 3′,5′‐MONOPHOSPHATE IN GUINEA PIG BRAIN 1

Only antihistaminic agents were capable of antagonizing the histamine‐induced increase of both [3H]‐ and total cyclic AMP in these two brain areas.
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