Dynamics of histamine H(3) receptor antagonists on brain histamine metabolism: do all histamine H(3) receptor antagonists act at a single site?

@article{Barnes2001DynamicsOH,
  title={Dynamics of histamine H(3) receptor antagonists on brain histamine metabolism: do all histamine H(3) receptor antagonists act at a single site?},
  author={William G. Barnes and D L Boyd and Lindsay B. Hough},
  journal={European journal of pharmacology},
  year={2001},
  volume={431 2},
  pages={
          215-21
        }
}
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Histamine turnover in regions of rat brain
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Results indicate that a potent and selective H3‐agonist, (R)‐α‐methylhistamine, and an H3-antagonist, thioperamide, have potent effects on HA turnover in vivo in the brain.
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