Design and synthesis of novel hydrocarbylidene nitrohydrazinecarboximidamides against aphids based on natural product galegine

  title={Design and synthesis of novel hydrocarbylidene nitrohydrazinecarboximidamides against aphids based on natural product galegine},
  author={Qinglai Wu and Fenghai Zhao and Xiang Zhu and Ziyuan Zhou and Dongyan Yang and Zhihong Xu and Jun-kai Li and Zhaohai Qin},
  journal={Natural Product Research},
  pages={1484 - 1490}
Abstract A series of novel hydrocarbylidene nitrohydrazinecarboximidamides were designed and synthesized using an insecticidal natural product Galegine as a lead compound. The bioassay results show that the target compounds exhibited moderate to good insecticidal activities against Hyalopterus pruni Geoffroy at a concentration of 200 mg/L, and most compounds show excellet insecticidal activities against Aphis gossypii Glover. In particular, compounds IIc-01, IIc-03, IIe-02 and IIf-01 show the… 

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