Corpus ID: 172036649

Derives de pyrazolo(1,5-a)pyridine utilises en tant que modulateurs du neurotransmetteur

@inproceedings{Fu2003DerivesDP,
  title={Derives de pyrazolo(1,5-a)pyridine utilises en tant que modulateurs du neurotransmetteur},
  author={Jianhao Fu},
  year={2003}
}
L'invention concerne des nouveaux derives de pyrazolo[1,5-a]pyridine representes par la formule generale (I), lesquels se lient avec une grande affinite aux recepteurs CRF1, y compris aux recepteurs CRF1 humains. La presente invention concerne egalement des methodes permettant d'utiliser ces composes pour traiter un trouble ou une affection pour lesquels le traitement peut etre realise ou facilite par antagonisation d'un recepteur CRF, tels que les maladies ou les troubles du systeme nerveux… Expand

References

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Based on the lead molecule FAUC 113, a series of di- and trisubstituted pyrazolo[1,5-a]pyridine derivatives was synthesized and investigated for their dopamine receptor binding profile. TheExpand
Synthesis of pyrazolo[1,5-a]pyridines and pyrazolo[1,5-c]pyrimidines by reaction of heterocyclic amidrazones with 1,3-dicarbonyl compounds
1,3-Dicarbonyl compounds 2 react with 1-amino-2(1H)-pyridin-2-imines or 1-amino-2(1H)-pyrimidin-2-imines 1 giving new pyrazolo[1,5-a]pyridines or pyrazolo[1,5-c]pyrimidines 5 respectively byExpand
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A convenient synthesis of derivatives of the pyrido[1′,2′:1,5]pyrazolo[3,4-d]pyrimidine ring system from readily available 2-amino-3-cyano-5,7-diphenylpyrazolo[1,5-a]pyridine I and carbon disulfide,Expand
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The syntheses and some reaetions of N,N'-diamino-2,2′- and 4,4′-bipyridinium salts (IV, V and VI) are described. These compounds are prepared by the reaction of bipyridyls (I-III) withExpand