Copper-catalyzed sequential N-arylation of C-amino-NH-azoles.

Abstract

Copper(II)-catalyzed boronic acid promoted C-N bond cross-coupling reactions have been successfully developed for sequential N-arylation of C-amino-NH-azoles. These general protocols are compatible with a variety of aryl/hetero-aryl boronic acids and provided rapid access to a diverse array of diarylaminoazole derivatives in a two-step sequence or in one… (More)
DOI: 10.1039/c4cc05628k

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@article{Rao2014CoppercatalyzedSN, title={Copper-catalyzed sequential N-arylation of C-amino-NH-azoles.}, author={Donthamsetty N Rao and S K Rasheed and Ram A Vishwakarma and Parthasarathi Das}, journal={Chemical communications}, year={2014}, volume={50 85}, pages={12911-4} }