Comparison of the effects of eleven histamine H1-receptor antagonists on monoamine turnover in the mouse brain

@article{Oishi2004ComparisonOT,
  title={Comparison of the effects of eleven histamine H1-receptor antagonists on monoamine turnover in the mouse brain},
  author={Ryozo Oishi and Setsu Shishido and Motoo Yamori and Kiyomi Saeki},
  journal={Naunyn-Schmiedeberg's Archives of Pharmacology},
  year={2004},
  volume={349},
  pages={140-144}
}
To compare in vivo effects of eleven compounds of different classes of histamine H1-receptor antagonists (alcoholamines: diphenhydramine, carbinoxamine, and clemastine; ethylenediamines: mepyramine, tripelennamine, and clemizole; alkylamines: triprolidine and chlorpheniramine; piperazines: meclizine and homochlorcyclizine; phenothiazines: promethazine) on neuronal uptake of dopamine (DA), noradrenaline (NA), and 5-hydroxytryptamine (5-HT), the effects on the turnover of these monoamines were… 
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Histamine and H3 receptor-dependent mechanisms regulate ethanol stimulation and conditioned place preference in mice
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Histaminergic neurotransmission seems to be necessary for the stimulatory effect of ethanol to occur, whereas lack of histamine leads to changes that enhance the conditioned reward by ethanol, suggesting a role for histamine H3 receptor in modulation of the ethanol stimulation and reward.
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