Comparison of 4-chloro-, 4-bromo- and 4-fluoroamphetamine in rats: Drug levels in brain and effects on brain serotonin metabolism
@article{Fuller1975ComparisonO4, title={Comparison of 4-chloro-, 4-bromo- and 4-fluoroamphetamine in rats: Drug levels in brain and effects on brain serotonin metabolism}, author={Ray W. Fuller and John C. Baker and Kenneth W. Perry and Bryan B. Molloy}, journal={Neuropharmacology}, year={1975}, volume={14}, pages={739-746} }
34 Citations
Studies on 4-(p-bromophenyl)-bicyclo (2,2,2) octan-1-amine as an inhibitor of uptake into serotonin neurones
- Biology, ChemistryNeuropharmacology
- 1978
5-hydroxytryptamine- and dopamine-releasing effects of ring-substituted amphetamines on rat brain: A comparative study using in vivo microdialysis
- Biology, ChemistryEuropean Neuropsychopharmacology
- 2014
Psychostimulant-like effects of p-fluoroamphetamine in the rat.
- Biology, ChemistryEuropean journal of pharmacology
- 1995
Para-halogenated phenethylamines: Similar serotonergic effects in rats by different mechanisms
- Chemistry, BiologyPharmacology Biochemistry and Behavior
- 1980
Effects of intraventricuear p-chloroamphetamine and its analogues on cerebral 5-HT
- Biology, ChemistryNeuropharmacology
- 1975
p-methylthioamphetamine is a potent new non-neurotoxic serotonin-releasing agent.
- Biology, ChemistryEuropean journal of pharmacology
- 1992
p-Chloroamphetamine (PCA), 3,4-methylenedioxymethamphetamine (MDMA) andd-fenfluramine pretreatment attenuatesd-fenfluramine-evoked release of 5-HT in vivo
- Biology, ChemistryPsychopharmacology
- 2005
The present data are consistent with the hypothesis that the acute release of 5-HT evoked by d-fenfluramine occurs via those terminals destroyed by pretreatment with PCA, MDMA andd-fen fluramine, while KCl evokes release from bothPCA-sensitive and PCA-insensitive terminals.
NEUROTOXIC ACTION OF HALOGENATED AMPHETAMINES *
- Biology, ChemistryAnnals of the New York Academy of Sciences
- 1978
Some of the anatomic evidence that has been obtained concerning the neurotoxic effects of various halogenated amphetamines by the use of Nissland silver-stained sections of brain are described.
Evaluation of nefopam as a monoamine uptake inhibitor in vivo in mice
- Biology, ChemistryNeuropharmacology
- 1993
A First-in-Man Study with 4-Fluoroamphetamine Demonstrates it Produces a Mild Psychedelic State
- PsychologyJournal of psychoactive drugs
- 2019
It is concluded that while the 4- FA-induced psychedelic state is mild in intensity and in between that produced by amphetamine and MDMA as hypothesized, more research is needed to indicate whether 4-FA can change creative thinking.
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