Comparative pharmacology of human β-adrenergic receptor subtypes—characterization of stably transfected receptors in CHO cells

@article{Hoffmann2003ComparativePO,
  title={Comparative pharmacology of human β-adrenergic receptor subtypes—characterization of stably transfected receptors in CHO cells},
  author={C. Hoffmann and M. Leitz and S. Oberdorf-Maass and M. Lohse and K. Klotz},
  journal={Naunyn-Schmiedeberg's Archives of Pharmacology},
  year={2003},
  volume={369},
  pages={151-159}
}
Although many β1-receptor antagonists and β2-receptor agonists have been used in pharmacotherapy for many years their pharmacological properties at all three known subtypes of β-adrenergic receptors are not always well characterized. The aim of this study was, therefore, to provide comparative binding characteristics of agonists (epinephrine, norepinephrine, isoproterenol, fenoterol, salbutamol, salmeterol, terbutalin, formoterol, broxaterol) and antagonists (propranolol, alprenolol, atenolol… Expand
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