CP-135,807, a selective 5-HT1D agonist: effects in drug discrimination and punishment procedures in the pigeon

@article{Mansbach1996CP135807AS,
  title={CP-135,807, a selective 5-HT1D agonist: effects in drug discrimination and punishment procedures in the pigeon},
  author={Robert S. Mansbach and Charles C. Rovetti and John Eugene Macor},
  journal={Psychopharmacology},
  year={1996},
  volume={128},
  pages={313-319}
}
Abstract CP-135,807 [3-(N-methylpyrrolidin-2R-ylmeth- yl)-5-(3-nitropyrid-2-yl)amino-1H-indole] binds with high affinity to central 5-HT1D receptors, and in functional studies produces dose-dependent decreases in extracellular serotonin. These and other findings have suggested that CP-135,807 may act as a terminal 5-HT autoreceptor agonist. In an attempt to characterize the behavioral activity of selective 5-HT1D ligands, adult male Carneau pigeons were trained to discriminate IM injections of… 

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