Binding selectivity of short [D-Arg2,Leu5]enkephalin analogues to mu- and delta-subclasses of opiate receptors.

Abstract

[D-Arg2,Leu5]enkephalin and its analogues, shortened from the C-terminus, were studied in a rat brain membrane fraction with the aid of radioreceptor analysis. The interaction between these compounds and the peripheral opiate receptors of isolated organs (guinea pig ileum and mouse vas deferens) was also investigated. The ethyl ester of the [D-Arg2… (More)

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@article{Rosenthal1990BindingSO, title={Binding selectivity of short [D-Arg2,Leu5]enkephalin analogues to mu- and delta-subclasses of opiate receptors.}, author={Gert Rosenthal and N M Inkina and N. A. Abissova and Irina Bobrova and Gunars Chipens}, journal={Biomedical science}, year={1990}, volume={1 4}, pages={414-6} }