Behavioral effects of (−)10, 11-methylenedioxy-n-n-propylnoraporphined, an orally effective long-acting agent active at central dopamine receptors, and analogous aporphines
@article{Campbell1982BehavioralEO, title={Behavioral effects of (−)10, 11-methylenedioxy-n-n-propylnoraporphined, an orally effective long-acting agent active at central dopamine receptors, and analogous aporphines}, author={Alexander Campbell and Ross J. Baldessarini and Vishnu Ji Ram and John L Neumeyer}, journal={Neuropharmacology}, year={1982}, volume={21}, pages={953-961} }
25 Citations
Tissue levels of N-n-propylnorapomorphine after treatment with (−)10,11-methylenedioxy-N-n-propylnoraporphine, an orally long-acting prodrug active at central dopamine receptors
- Biology, ChemistryNeuropharmacology
- 1982
S(+)methylenedioxy-N-n-propylnoraporphine: an orally active inhibitor of dopamine selective for rat limbic system
- Biology, PsychologyBrain Research
- 1987
Behavioral effects of apomorphine isomers in the rat: Selective locomotor-inhibitory effects of S(+)N-n-propylnorapomorphine
- Biology, PsychologyPsychopharmacology
- 2004
The results suggest that S(+)NPA or its congeners and analogs may have selective antidopaminergic actions in limbic rather than striatal areas of mammalian brain.
Behavioral activity of some novel aporphines in rats with 6-hydroxydopamine lesions of caudate or nucleus accumbens.
- Biology, PsychologyEuropean journal of pharmacology
- 1983
Striatally-mediated response of some structurally rigid analogues of dopamine
- Chemistry, BiologyPharmacology Biochemistry and Behavior
- 1986
Prolonged antidopaminergic actions of single doses of butyrophenones in the rat
- Psychology, BiologyPsychopharmacology
- 2004
The results indicate that some neuroleptics may have very prolonged activity or retention in tissue at sites of action, even after moderate, single doses.
Synthesis and neuropharmacological evaluation of R(-)-N-alkyl-11-hydroxynoraporphines and their esters.
- Biology, ChemistryBioorganic & medicinal chemistry
- 2004
S(+)apomorphines selective inhibition of excitatory effects of dopamine injected into the limbic system of the rat
- Biology, PsychologyNeuropharmacology
- 1985
Comparative assessment of dopamine agonist aporphines as anticonvulsants in two models of reflex epilepsy
- Chemistry, MedicinePsychopharmacology
- 2004
All the compounds (including norapomorphine) significantly lowered rectal temperature, although the time course of this effect was often longer than that of protection against audiogenic seizures.
Effect of age on behavioral responses and tissue levels of apomorphine in the rat
- Biology, PsychologyNeuropharmacology
- 1984
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