Corpus ID: 34274461

Antitumor activity of homo-aza-steroidal esters of p-N, N-bis(2-chloroethyl)aminophenoxyacetic acid.

@article{Catsoulacos1993AntitumorAO,
  title={Antitumor activity of homo-aza-steroidal esters of p-N, N-bis(2-chloroethyl)aminophenoxyacetic acid.},
  author={P. Catsoulacos and D. Catsoulacos},
  journal={Anticancer research},
  year={1993},
  volume={13 4},
  pages={
          1203-8
        }
}
  • P. Catsoulacos, D. Catsoulacos
  • Published 1993
  • Chemistry, Medicine
  • Anticancer research
    • The homo-aza-steroidal esters of carboxylic derivatives of N, N-bis (2-chloroethyl) aniline are reviewed. In particular, we discuss the antitumor activity of the esters of homo-aza steroids in which the p-N,N-bis(2-chloroethyl)aminophenoxyacetic acid is linked to the C-3 or C-17 position, while the lactam nucleus is linked to the D or A ring of the modified steroid respectively. The current literature indicates clearly that the potential of these esters is due to the synergistic activity of… CONTINUE READING
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