An improved one-pot method for the stereoselective synthesis of the (2S,3R)-3-amino-2-hydroxy acids: key intermediates for bestatin and amastatin

@article{Herranz1990AnIO,
  title={An improved one-pot method for the stereoselective synthesis of the (2S,3R)-3-amino-2-hydroxy acids: key intermediates for bestatin and amastatin},
  author={Rosario Herranz and Julia Castro‐Pichel and Soledad Vinuesa and Ma Teresa Garc{\'i}a-L{\'o}pez},
  journal={Journal of Organic Chemistry},
  year={1990},
  volume={55},
  pages={2232-2234}
}
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59 Citations
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Facile Synthesis of (2S,3R)-3-Amino-2-Hydroxycarboxylic Acids, the Key Components of Amastatin and Bestatin
Abstract The title amino acids, (2S,3R)-3-amino-2-hydroxy-5-methyl-hexanoic acid (AHMHA) and (2S,3R)-3-amino-2-hydroxy-4-phenylbutanoic acid (AHPBA), are stereoselectively prepared from
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