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Drug discovery targeting amino acid racemases.
- P. Conti, L. Tamborini, C. De Micheli
- Chemistry, MedicineChemical reviews
- 13 September 2011
Drug Discovery Targeting Amino Acid Racemases Paola Conti, Lucia Tamborini, Andrea Pinto, Arnaud Blondel, Paola Minoprio, Andrea Mozzarelli, and Carlo De Micheli* Dipartimento di Scienze…
Design of remarkably simple, yet potent urea-based inhibitors of glutamate carboxypeptidase II (NAALADase).
- A. Kozikowski, F. Nan, J. Wroblewski
- BiologyJournal of medicinal chemistry
- 3 January 2001
Synthesis and biochemical evaluation of δ(2)-isoxazoline derivatives as DNA methyltransferase 1 inhibitors.
- S. Castellano, D. Kuck, G. Sbardella
- Chemistry, BiologyJournal of medicinal chemistry
- 1 September 2010
A series of Δ(2)-isoxazoline constrained analogues of procaine/procainamide (7a-k and 8a-k) were prepared and their inhibitory activity against DNA methyltransferase 1 (DNMT1) was tested. Among them,…
The Glial Glutamate Transporter 1 (GLT1) Is Expressed by Pancreatic β-Cells and Prevents Glutamate-induced β-Cell Death*
- E. D. Di Cairano, A. Davalli, C. Perego
- BiologyThe Journal of Biological Chemistry
- 18 February 2011
TLDR
Mutant p53 prevents GAPDH nuclear translocation in pancreatic cancer cells favoring glycolysis and 2-deoxyglucose sensitivity.
- Giovanna Butera, R. Pacchiana, M. Donadelli
- BiologyBiochimica et biophysica acta. Molecular cell…
- 1 December 2018
Marine Microorganisms as Source of Stereoselective Esterases and Ketoreductases: Kinetic Resolution of a Prostaglandin Intermediate
TLDR
Synthesis of (3-hydroxy-pyrazolin-5-yl)glycine based ligands interacting with ionotropic glutamate receptors.
- A. Pinto, L. Tamborini, P. Conti
- Chemistry, BiologyEuropean journal of medicinal chemistry
- 21 March 2014
Inspired by Nature: The 3‐Halo‐4,5‐dihydroisoxazole Moiety as a Novel Molecular Warhead for the Design of Covalent Inhibitors
- A. Pinto, L. Tamborini, Gregorio Cullia, P. Conti, C. De Micheli
- Chemistry, BiologyChemMedChem
- 2016
TLDR
Synthesis and functional characterization of novel derivatives related to oxotremorine and oxotremorine-M.
- C. Dallanoce, P. Conti, M. Impicciatore
- Biology, ChemistryBioorganic & medicinal chemistry
- 1 August 1999
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