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One pot, Solvent-free synthesis of substituted 3,4-dihydropyrimidin- 2(1H)-ones/thiones under microwave irradiation (CEM) using reusable nickel nanoparticles
A library of 3,4-dihydropyrimidin-2(1H)-ones/thiones derivatives were synthesized via Biginelli condensation reaction of β-keto esters, aryl aldehydes and urea/thiourea under solvent-free conditions…
Pyrimidine‐based pyrazoles as cyclin‐dependent kinase 2 inhibitors: Design, synthesis, and biological evaluation
- Mayur K. Vekariya, Rajesh H. Vekariya, P. Brahmkshatriya, N. Shah
- Chemistry, MedicineChemical biology & drug design
- 19 June 2018
It is shown that of the 26 compounds synthesized and evaluated, at least 5 compounds were found to be highly potent (IC50 < 20 nm); which can be further optimized to have selectivity over other kinase isoforms.
Microwave-assisted green synthesis of new imidazo[2,1-b]thiazole derivatives and their antimicrobial, antimalarial, and antitubercular activities
- Rajesh H. Vekariya, K. Patel, +4 authors H. Patel
- ChemistryResearch on Chemical Intermediates
- 22 May 2017
We have synthesized some imidazo[2,1-b]thiazole derivatives by reaction of 1-(2-amino-4-methylthiazol-5-yl)ethanone or ethyl 2-amino-4-methylthiazole-5-carboxylate with α-bromo aralkyl ketones…
Pyrimidine-Pyrazole Hybrids as Morpholinopyrimidine-Based Pyrazole Carboxamides: Synthesis, Characterisation, Docking, ADMET Study and Biological Evaluation
Novel N-thioamide analogues of pyrazolylpyrimidine based piperazine: Design, synthesis, characterization, in-silico molecular docking study and biological evaluation
Synthesis, characterization and adsorption significance of novel composite (chitosan beads loaded nickel-oxide nanoparticles)
Preparation of α-Iodocarbonyl Compounds: An Overall Development
Adsorption of lead (II) ions onto novel cassava starch 5-choloromethyl-8-hydroxyquinoline polymer from an aqueous medium.
- Prapti U. Shah, Nirav P. Raval, Mayur K. Vekariya, P. Wadhwani, N. Shah
- Chemistry, MedicineWater science and technology : a journal of the…
- 17 August 2016
The results indicate that CSCMQ could be employed as low-cost material for the adsorption of Pb(II) ions from aqueous medium.
Synthesis of pyrazolo[4ʹ,3ʹ:5,6]pyrano[2,3- d ]pyrimidine derivatives and their antimicrobial, antimalarial and antituberculosis evaluation
This article deals with the synthesis of a new pyrazolo[4ʹ,3ʹ:5,6]pyrano[2,3-d]pyrimidine derivatives by the reaction of 1,4-dihydropyrano[2,3-c]-pyrazole-5-carbonitriles with ethyl cyanoacetate…
Green synthesis of pyrazolo[4,3- d ]isoxazol derivatives and their antimicrobial, antimalarial and antituberculosis evaluation
This article deals with the synthesis of new pyrazolo[4,3-d]isoxazol derivatives by utilizing 3,4-disubstituted isoxazol5(4H)-ones and thiosemicarbazide catalyzed by triethylamine in PEG-400 under…